Drug classDrugDosagesComplications
Estrogen antagonistsTamoxifen (Nolvadex)20 mg per dayHot flushes, drying of vaginal secretions, deep venous thrombosis, retinopathy, hypercalcemia*
ProgestinsMegestrol (Megace)40 mg four times dailyWeight gain, nausea, fluid retention
Aromatase inhibitorsAminoglutethimide (Cytadren)250 mg twice dailySomnolence, skin rash, hypoadrenalism
Anastrozole (Arimidex)1 mg per dayNone
Letrozole (Femara)50 mg (one tablet) per dayNone
EstrogensDiethylstilbestrol5 mg three times dailyDeep venous thrombosis, fluid retention, hypercalcemia*
AndrogensFluoxymesterone (Halotestin)10 mg three times dailyVirilization, fluid retention