Estrogen antagonists | Tamoxifen (Nolvadex) | 20 mg per day | Hot flushes, drying of vaginal secretions, deep venous thrombosis, retinopathy, hypercalcemia* |
Progestins | Megestrol (Megace) | 40 mg four times daily | Weight gain, nausea, fluid retention |
Aromatase inhibitors | Aminoglutethimide (Cytadren)† | 250 mg twice daily | Somnolence, skin rash, hypoadrenalism |
Anastrozole (Arimidex) | 1 mg per day | None |
Letrozole (Femara) | 50 mg (one tablet) per day | None |
Estrogens | Diethylstilbestrol | 5 mg three times daily | Deep venous thrombosis, fluid retention, hypercalcemia* |
Androgens | Fluoxymesterone (Halotestin) | 10 mg three times daily | Virilization, fluid retention |